根皮素

分析標(biāo)準(zhǔn)品,HPLC≥98%

Phloretin

CAS號(hào)：60-82-2

分子式：C15H14O5

分子量：274.27

MDL：MFCD00002288

別名：2',4',6'-三羥基-3-(4-羥基苯基)苯丙酮;3-(4-羥苯基)-1-(2,4,6-三羥基苯基)-1-丙酮

產(chǎn)品介紹

根皮素  Phloretin (NSC 407292; RJC 02792) 是一種從蘋果中提取的黃酮類化合物，具有抗炎活性。Phloridzin 是一種特異性、競(jìng)爭(zhēng)性和口服活性的鈉/葡萄糖協(xié)同轉(zhuǎn)運(yùn)蛋白 (sodium/glucose cotransporters) 抑制劑，在腸道 (SGLT1) 和腎臟 (SGLT2)。Phloretin 抑制 Yeast-made GLUT1 以及人類紅細(xì)胞 GLUT1 的 IC50 值分別為 49 μM 和 61 μM。Phloretin 具有潛力用于類風(fēng)濕性關(guān)節(jié)炎 (RA) 和過(guò)敏性氣道炎癥的相關(guān)研究。

熔點(diǎn)：260-262℃

沸點(diǎn)：534.4 ℃ at 760 mmHg

外觀：淡紅色粉末狀

溶解性：DMSO:50mg/mL(182.30mM;Need ultrasonic)

H2O:0.1mg/mL(0.36mM;Need ultrasonic)

敏感性：對(duì)熱和光敏感

儲(chǔ)存條件：-20℃

注意：部分產(chǎn)品我司僅能提供部分信息，我司不保證所提供信息的權(quán)威性，僅供客戶參考交流研究之用。

參考文獻(xiàn)(56篇)

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