大黃素甲醚

分析標準品,HPLC≥98%

Physcion

CAS號：521-61-9

分子式：C16H12O5

分子量：284.26

MDL：MFCD00017374

產(chǎn)品介紹

Physcion (Parietin) 是從中藥大黃中得到的蒽醌類物質(zhì)，為 6-磷酸葡萄糖酸脫氫酶 (6-phosphogluconate dehydrogenase) 抑制劑，IC50 和 Kd 值分別為 38.5 μM 和 26.0 μM。Physcion (Parietin) 具有通便、保肝、抗炎、抗菌、抗增殖、抗腫瘤作用。

熔點：196-206℃

沸點：560.5℃ at 760 mmHg

外觀：黃色結(jié)晶

溶解性：DMSO : 3.33mg/mL(11.71mM;ultrasonicandwarming and adjust pH to 9withNaOH and heat to 60℃)

THF :2.5mg/mL(8.79mM; ultrasonic and warming and heat to 60℃)

DMF : 1mg/mL(3.52mM;Needultrasonic)

Acetone : < 1mg/mL(insoluble)

Methanol :< 1mg/mL(ultrasonic)(insoluble)

Ethanol : < 1mg/mL(insoluble)

儲存條件：2-8℃

注意：部分產(chǎn)品我司僅能提供部分信息，我司不保證所提供信息的權(quán)威性，僅供客戶參考交流研究之用。

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